├── .gitignore
├── .idea
├── .gitignore
├── SAMPL8.iml
├── inspectionProfiles
│ └── profiles_settings.xml
├── misc.xml
├── modules.xml
├── other.xml
├── rGraphicsSettings.xml
├── rSettings.xml
└── vcs.xml
├── LICENSE
├── LICENSE_other
├── README.md
├── host_guest
├── Analysis
│ ├── All_Accuracy
│ │ ├── CB8
│ │ │ ├── EnthalpiesCorrelationPlots
│ │ │ │ ├── 14.pdf
│ │ │ │ ├── 30.pdf
│ │ │ │ └── 6.pdf
│ │ │ ├── FreeEnergyCorrelationPlots
│ │ │ │ ├── 1.pdf
│ │ │ │ ├── 10.pdf
│ │ │ │ ├── 11.pdf
│ │ │ │ ├── 12.pdf
│ │ │ │ ├── 13.pdf
│ │ │ │ ├── 14.pdf
│ │ │ │ ├── 15.pdf
│ │ │ │ ├── 16.pdf
│ │ │ │ ├── 17.pdf
│ │ │ │ ├── 18.pdf
│ │ │ │ ├── 19.pdf
│ │ │ │ ├── 2.pdf
│ │ │ │ ├── 20.pdf
│ │ │ │ ├── 21.pdf
│ │ │ │ ├── 22.pdf
│ │ │ │ ├── 23.pdf
│ │ │ │ ├── 24.pdf
│ │ │ │ ├── 25.pdf
│ │ │ │ ├── 26.pdf
│ │ │ │ ├── 27.pdf
│ │ │ │ ├── 28.pdf
│ │ │ │ ├── 29.pdf
│ │ │ │ ├── 3.pdf
│ │ │ │ ├── 30.pdf
│ │ │ │ ├── 31.pdf
│ │ │ │ ├── 32.pdf
│ │ │ │ ├── 33.pdf
│ │ │ │ ├── 34.pdf
│ │ │ │ ├── 4.pdf
│ │ │ │ ├── 5.pdf
│ │ │ │ ├── 6.pdf
│ │ │ │ ├── 7.pdf
│ │ │ │ ├── 8.pdf
│ │ │ │ └── 9.pdf
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ ├── R2_bootstrap_distributions.pdf
│ │ │ │ ├── RMSE_bootstrap_distributions.pdf
│ │ │ │ ├── kendall_tau_bootstrap_distributions.pdf
│ │ │ │ └── m_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ └── bootstrap_distributions.p
│ │ ├── GDCC
│ │ │ ├── FreeEnergyCorrelationPlots
│ │ │ │ ├── 35.pdf
│ │ │ │ ├── 36.pdf
│ │ │ │ ├── 37.pdf
│ │ │ │ ├── 38.pdf
│ │ │ │ ├── 39.pdf
│ │ │ │ ├── 40.pdf
│ │ │ │ ├── 41.pdf
│ │ │ │ ├── 42.pdf
│ │ │ │ ├── 43.pdf
│ │ │ │ ├── 44.pdf
│ │ │ │ ├── 45.pdf
│ │ │ │ ├── 46.pdf
│ │ │ │ ├── 47.pdf
│ │ │ │ ├── 48.pdf
│ │ │ │ ├── 49.pdf
│ │ │ │ ├── 50.pdf
│ │ │ │ └── 51.pdf
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ ├── R2_bootstrap_distributions.pdf
│ │ │ │ ├── RMSE_bootstrap_distributions.pdf
│ │ │ │ ├── kendall_tau_bootstrap_distributions.pdf
│ │ │ │ └── m_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ └── bootstrap_distributions.p
│ │ ├── GDCC_no_optional
│ │ │ ├── FreeEnergyCorrelationPlots
│ │ │ │ ├── 35.pdf
│ │ │ │ ├── 36.pdf
│ │ │ │ ├── 37.pdf
│ │ │ │ ├── 38.pdf
│ │ │ │ ├── 39.pdf
│ │ │ │ ├── 40.pdf
│ │ │ │ ├── 41.pdf
│ │ │ │ ├── 42.pdf
│ │ │ │ ├── 43.pdf
│ │ │ │ ├── 44.pdf
│ │ │ │ ├── 45.pdf
│ │ │ │ ├── 46.pdf
│ │ │ │ ├── 47.pdf
│ │ │ │ ├── 48.pdf
│ │ │ │ ├── 49.pdf
│ │ │ │ ├── 50.pdf
│ │ │ │ └── 51.pdf
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ ├── R2_bootstrap_distributions.pdf
│ │ │ │ ├── RMSE_bootstrap_distributions.pdf
│ │ │ │ ├── kendall_tau_bootstrap_distributions.pdf
│ │ │ │ └── m_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ └── bootstrap_distributions.p
│ │ ├── MoleculesStatistics
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ └── RMSE_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ ├── bootstrap_distributions.p
│ │ │ └── molecules_error.pdf
│ │ ├── PaperImages
│ │ │ └── error_by_molecule.pdf
│ │ └── README.md
│ ├── ExperimentalMeasurements
│ │ ├── CB8-DOA-SAMPL-Answer-Sheet-20201014.docx
│ │ ├── CB8-DOA-SAMPL-Answer-Sheet-20201014.pdf
│ │ ├── Final-Data-Table-031621-SAMPL8.docx
│ │ ├── PDFTable
│ │ │ ├── experimental_measurements.pdf
│ │ │ └── experimental_measurements.tex
│ │ ├── README.md
│ │ ├── experimental_measurements.csv
│ │ ├── experimental_measurements.json
│ │ └── generate_tables.py
│ ├── README.md
│ ├── Ranked_Accuracy
│ │ ├── CB8
│ │ │ ├── EnthalpiesCorrelationPlots
│ │ │ │ ├── 30.pdf
│ │ │ │ └── 6.pdf
│ │ │ ├── FreeEnergyCorrelationPlots
│ │ │ │ ├── 1.pdf
│ │ │ │ ├── 11.pdf
│ │ │ │ ├── 13.pdf
│ │ │ │ ├── 15.pdf
│ │ │ │ ├── 2.pdf
│ │ │ │ ├── 28.pdf
│ │ │ │ ├── 3.pdf
│ │ │ │ ├── 30.pdf
│ │ │ │ ├── 6.pdf
│ │ │ │ └── 7.pdf
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ ├── R2_bootstrap_distributions.pdf
│ │ │ │ ├── RMSE_bootstrap_distributions.pdf
│ │ │ │ ├── kendall_tau_bootstrap_distributions.pdf
│ │ │ │ └── m_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ └── bootstrap_distributions.p
│ │ ├── GDCC
│ │ │ ├── FreeEnergyCorrelationPlots
│ │ │ │ ├── 36.pdf
│ │ │ │ ├── 37.pdf
│ │ │ │ ├── 38.pdf
│ │ │ │ ├── 39.pdf
│ │ │ │ ├── 43.pdf
│ │ │ │ ├── 44.pdf
│ │ │ │ ├── 45.pdf
│ │ │ │ └── 46.pdf
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ ├── R2_bootstrap_distributions.pdf
│ │ │ │ ├── RMSE_bootstrap_distributions.pdf
│ │ │ │ ├── kendall_tau_bootstrap_distributions.pdf
│ │ │ │ └── m_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ └── bootstrap_distributions.p
│ │ ├── GDCC_no_optional
│ │ │ ├── FreeEnergyCorrelationPlots
│ │ │ │ ├── 36.pdf
│ │ │ │ ├── 37.pdf
│ │ │ │ ├── 38.pdf
│ │ │ │ ├── 39.pdf
│ │ │ │ ├── 43.pdf
│ │ │ │ ├── 44.pdf
│ │ │ │ ├── 45.pdf
│ │ │ │ └── 46.pdf
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ ├── R2_bootstrap_distributions.pdf
│ │ │ │ ├── RMSE_bootstrap_distributions.pdf
│ │ │ │ ├── kendall_tau_bootstrap_distributions.pdf
│ │ │ │ └── m_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ └── bootstrap_distributions.p
│ │ ├── MoleculesStatistics
│ │ │ ├── StatisticsPlots
│ │ │ │ ├── MAE_bootstrap_distributions.pdf
│ │ │ │ ├── ME_bootstrap_distributions.pdf
│ │ │ │ └── RMSE_bootstrap_distributions.pdf
│ │ │ ├── StatisticsTables
│ │ │ │ ├── statistics.csv
│ │ │ │ ├── statistics.json
│ │ │ │ └── statisticsLaTex
│ │ │ │ │ └── statistics.tex
│ │ │ ├── bootstrap_distributions.p
│ │ │ └── molecules_error.pdf
│ │ ├── PaperImages
│ │ │ ├── Figure2_experimental_measurements.pdf
│ │ │ ├── Figure_correlation_plots_ranked_methods.pdf
│ │ │ ├── error_by_molecule.pdf
│ │ │ └── tightest_binders.pdf
│ │ └── README.md
│ ├── SAMPL8-user-map-HG.csv
│ ├── Scripts
│ │ ├── README.md
│ │ ├── analyze_hostguest.py
│ │ ├── get_usermap.py
│ │ ├── pkganalysis
│ │ │ ├── __init__.py
│ │ │ ├── stats.py
│ │ │ └── submission.py
│ │ └── update_usermap.py
│ └── Submissions
│ │ ├── CB8
│ │ ├── CB8-Hansen-1.txt
│ │ ├── CB8-Hansen-2.txt
│ │ ├── CB8-sampl8-submission-LiGaMD.txt
│ │ ├── CB8_MahdiGhorbani.txt
│ │ ├── CB8_NIH0.txt
│ │ ├── CB8_NIH1.txt
│ │ ├── CB8_NIH10.txt
│ │ ├── CB8_NIH11.txt
│ │ ├── CB8_NIH12.txt
│ │ ├── CB8_NIH2.txt
│ │ ├── CB8_NIH3.txt
│ │ ├── CB8_NIH4.txt
│ │ ├── CB8_NIH5.txt
│ │ ├── CB8_NIH6.txt
│ │ ├── CB8_NIH7.txt
│ │ ├── CB8_NIH8.txt
│ │ ├── CB8_NIH9.txt
│ │ ├── CB8_REF_GAFF2_MBAR.txt
│ │ ├── CB8_REF_GAFF2_TI.txt
│ │ ├── CB8_REF_OPENFF_MBAR.txt
│ │ ├── CB8_REF_OPENFF_TI.txt
│ │ ├── CB8_SILCS_rawLGFE.txt
│ │ ├── CB8_SILCS_rawLGFE_G5.txt
│ │ ├── CB8_SILCS_reweightedLGFE.txt
│ │ ├── CB8_Selim_BigginLab.txt
│ │ ├── CB8_Selim_BigginLab_Ranked.txt
│ │ ├── CB8_Submission.txt
│ │ ├── CB8_dserillon_CB8MLs_UNRANKED.txt
│ │ ├── CB8_dserillon_GlobalisticMLs_UNRANKED.txt
│ │ ├── CB8_dserillon_PhysicBasedMethod_BA_UNRANKED.txt
│ │ ├── CB8_dserillon_PhysicBasedMethod_RANKED.txt
│ │ ├── CB8_fm3_lw.txt
│ │ ├── CB8_submission_ARNOLD.txt
│ │ ├── CB8_submissions.txt
│ │ ├── CB8_template
│ │ └── submission_file_converter.ipynb
│ │ ├── GDCC
│ │ ├── GDCC-ATM.txt
│ │ ├── GDCC-PMF.txt
│ │ ├── GDCC-ponder.txt
│ │ ├── GDCC_GAFF2_MBAR.txt
│ │ ├── GDCC_GAFF2_TI.txt
│ │ ├── GDCC_GlobalisticML_dserillon.txt
│ │ ├── GDCC_LCB.txt
│ │ ├── GDCC_MahdiGhorbani.txt.txt
│ │ ├── GDCC_PBSA_AM1BCC_nonranked.txt
│ │ ├── GDCC_PBSA_AM1BCC_nonranked_2020S6OA.txt
│ │ ├── GDCC_PBSA_AM1BCC_nonranked_2020S6OA_3Vd1WFL.txt
│ │ ├── GDCC_PBSA_AM1BCC_ranked_2c.txt
│ │ ├── GDCC_Parsley_MBAR.txt
│ │ ├── GDCC_Parsley_TI.txt
│ │ ├── GDCC_SILCS_rawLGFE.txt
│ │ ├── GDCC_SILCS_reweightedLGFE.txt
│ │ └── GDCC_submissions-LiGaMD.txt
│ │ └── README.md
├── CB8
│ ├── CB8_submissions.txt
│ ├── README.md
│ ├── guest_files
│ │ ├── CB8_guest_names.txt
│ │ ├── CB8_guest_smiles.txt
│ │ ├── G1.mol2
│ │ ├── G1.pdb
│ │ ├── G1.sdf
│ │ ├── G2.mol2
│ │ ├── G2.pdb
│ │ ├── G2.sdf
│ │ ├── G3.mol2
│ │ ├── G3.pdb
│ │ ├── G3.sdf
│ │ ├── G4.mol2
│ │ ├── G4.pdb
│ │ ├── G4.sdf
│ │ ├── G5.mol2
│ │ ├── G5.pdb
│ │ ├── G5.sdf
│ │ ├── G6.mol2
│ │ ├── G6.pdb
│ │ ├── G6.sdf
│ │ ├── G7.mol2
│ │ ├── G7.pdb
│ │ ├── G7.sdf
│ │ ├── README.md
│ │ └── input_maker.ipynb
│ ├── host_files
│ │ ├── Assign_Charge.ipynb
│ │ ├── CB8.mol2
│ │ ├── CB8.pdb
│ │ ├── CB8.sdf
│ │ └── README.md
│ ├── images
│ │ └── CB8_overview.png
│ └── source_files
│ │ ├── CB8_chemdraw.cdx
│ │ ├── README.md
│ │ ├── description.docx
│ │ ├── description.pdf
│ │ └── ~$scription.docx
├── GDCC
│ ├── GDCC_submissions.txt
│ ├── Hosts.png
│ ├── README.md
│ ├── guest_files
│ │ ├── G1.mol2
│ │ ├── G1.pdb
│ │ ├── G1.sdf
│ │ ├── G2.mol2
│ │ ├── G2.pdb
│ │ ├── G2.sdf
│ │ ├── G3.mol2
│ │ ├── G3.pdb
│ │ ├── G3.sdf
│ │ ├── G4.mol2
│ │ ├── G4.pdb
│ │ ├── G4.sdf
│ │ ├── G5.mol2
│ │ ├── G5.pdb
│ │ ├── G5.sdf
│ │ ├── README.md
│ │ ├── guest_smiles.csv
│ │ └── guest_smiles.txt
│ ├── guests.cdx
│ ├── guests.pdf
│ ├── guests.png
│ ├── host_files
│ │ ├── Assign_Charge.ipynb
│ │ ├── README.md
│ │ ├── TEEtOA.mol2
│ │ ├── TEEtOA.pdb
│ │ ├── TEEtOA.sdf
│ │ ├── TEEtOA_charge.mol2
│ │ ├── TEMOA.mol2
│ │ ├── TEMOA.pdb
│ │ ├── TEMOA.sdf
│ │ └── TEMOA_charge.mol2
│ ├── input_maker.ipynb
│ └── source_files
│ │ ├── .DS_Store
│ │ ├── Compound Identifiers.xlsx
│ │ ├── Guests
│ │ ├── .DS_Store
│ │ ├── 3-hydroxy-2-naphthoic acid
│ │ │ ├── 3-hydroxy-2-naphthoic acid.cdx
│ │ │ ├── 3-hydroxy-2-naphthoic acid.mol2
│ │ │ ├── 3-hydroxy-2-naphthoic acid.pdb
│ │ │ └── 3-hydroxy-2-naphthoic acid.sdf
│ │ ├── 4-Bromophenol
│ │ │ ├── 4-bromophenol.cdx
│ │ │ ├── 4-bromophenol.mol2
│ │ │ ├── 4-bromophenol.pdb
│ │ │ └── 4-bromophenol.sdf
│ │ ├── Cyclopentylacetic acid
│ │ │ ├── Cyclopentylacetic acid.cdx
│ │ │ ├── cyclopentylacetic acid.mol2
│ │ │ ├── cyclopentylacetic acid.pdb
│ │ │ └── cyclopentylacetic acid.sdf
│ │ ├── Piperonylic acid
│ │ │ ├── piperonylic acid.cdx
│ │ │ ├── piperonylic acid.mol2
│ │ │ ├── piperonylic acid.pdb
│ │ │ └── piperonylic acid.sdf
│ │ └── p-toluic acid
│ │ │ ├── p-toluic acid.cdx
│ │ │ ├── p-toluic acid.mol2
│ │ │ ├── p-toluic acid.pdb
│ │ │ └── p-toluic acid.sdf
│ │ ├── Hosts.tiff
│ │ ├── Hosts
│ │ ├── TEEtOA
│ │ │ ├── TEEtOA.cdx
│ │ │ ├── TEEtOA.mol2
│ │ │ ├── TEEtOA.pdb
│ │ │ └── TEEtOA.sdf
│ │ └── TEMOA
│ │ │ ├── TEMOA.cdx
│ │ │ ├── TEMOA.mol2
│ │ │ ├── TEMOA.pdb
│ │ │ └── TEMOA.sdf
│ │ └── README.md
├── README.md
└── Scripts
│ ├── get_usermap.py
│ └── make_guest_iupac_names.py
├── host_guest_instructions.md
└── physical_properties
├── README.md
├── SAMPL8_molecule_ID_and_SMILES.csv
├── experimental_data
├── Aqueous_Solubility for SAMPL8 Pub.xlsx
├── Log D Summary Calculations Final MNB Pub.xls
├── README.md
├── SAMPL Structures from SMILES.xlsx
├── SAMPL8 - SiriusT3 measurements.pdf
├── SAMPL8 Final Readout_Distribution Coefficient Pub.pptx
├── SAMPL8 Final Readout_pH-Solubility Pub.pptx
├── pKa - SiriusT3 measurements.csv
└── pKa.csv
├── images
├── SAMPL8-molecules.pdf
├── SAMPL8-molecules.png
└── SAMPL8-molecules.svg
├── logD
├── README.md
├── SAMPL8-logD-user-map.csv
├── SAMPL8-logD_experimental_values.csv
├── analysis
│ ├── README.md
│ ├── Submissions
│ │ ├── logD-3DS-1.csv
│ │ ├── logD-AndreaEbert-1_tF851UO.csv
│ │ ├── logD-ECRISM-1.csv
│ │ ├── logD-ECRISM-2.csv
│ │ ├── logD-ECRISM-3.csv
│ │ ├── logD-IEFPCMMST-1.csv
│ │ ├── logD-IEFPCMMST-2.csv
│ │ ├── logD-NadinUlrich-1.csv
│ │ ├── logD-NadinUlrich-1_9C8eUz5.csv
│ │ ├── logD-UCRMLR0-5.csv
│ │ ├── logD-UCRMLR0-6.csv
│ │ ├── logD-UCRMLR06-7.csv
│ │ ├── logD-UCRMLR06-8.csv
│ │ ├── logD-UCRPLS3-1.csv
│ │ ├── logD-UCRPLS3-2.csv
│ │ ├── logD-UCRPLS3-2_gplfkzn.csv
│ │ ├── logD-UCRPLS3REL-3.csv
│ │ ├── logD-UCRPLS3REL-4.csv
│ │ ├── logD-ZhiyiWu-1.csv
│ │ ├── logD-davyguan-1.csv
│ │ ├── logD_OllierTranPaluch_LSER_exp.csv
│ │ ├── logD_OllierTranPaluch_UFZ_LSER_exp.csv
│ │ ├── logD_SAMPL8_ShuzheWang_ranked.csv
│ │ ├── logD_SAMPL8_ShuzheWang_unranked1.csv
│ │ ├── logD_SAMPL8_ShuzheWang_unranked2.csv
│ │ ├── logD_SAMPL8_ShuzheWang_unranked3.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_2.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_3.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_2.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_3.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_extra.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_extra_2.csv
│ │ └── logD_SabatinoRodriguezPaluch_uESE_extra_3.csv
│ ├── Submissions_edited
│ │ ├── logD-3DS-1.csv
│ │ ├── logD-AndreaEbert-1_tF851UO.csv
│ │ ├── logD-ECRISM-1.csv
│ │ ├── logD-ECRISM-2.csv
│ │ ├── logD-ECRISM-3.csv
│ │ ├── logD-IEFPCMMST-1.csv
│ │ ├── logD-IEFPCMMST-2.csv
│ │ ├── logD-NadinUlrich-1.csv
│ │ ├── logD-NadinUlrich-1_9C8eUz5.csv
│ │ ├── logD-UCRMLR0-5.csv
│ │ ├── logD-UCRMLR0-6.csv
│ │ ├── logD-UCRMLR06-7.csv
│ │ ├── logD-UCRMLR06-8.csv
│ │ ├── logD-UCRPLS3-1.csv
│ │ ├── logD-UCRPLS3-2.csv
│ │ ├── logD-UCRPLS3-2_gplfkzn.csv
│ │ ├── logD-UCRPLS3REL-3.csv
│ │ ├── logD-UCRPLS3REL-4.csv
│ │ ├── logD-ZhiyiWu-1.csv
│ │ ├── logD-davyguan-1.csv
│ │ ├── logD_OllierTranPaluch_LSER_exp.csv
│ │ ├── logD_OllierTranPaluch_UFZ_LSER_exp.csv
│ │ ├── logD_SAMPL8_ShuzheWang_ranked.csv
│ │ ├── logD_SAMPL8_ShuzheWang_unranked1.csv
│ │ ├── logD_SAMPL8_ShuzheWang_unranked2.csv
│ │ ├── logD_SAMPL8_ShuzheWang_unranked3.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_2.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_3.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_2.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_3.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_extra.csv
│ │ ├── logD_SabatinoRodriguezPaluch_uESE_extra_2.csv
│ │ └── logD_SabatinoRodriguezPaluch_uESE_extra_3.csv
│ ├── analysis_all
│ │ ├── Performance_stats_by_solvent_combo
│ │ │ └── Error_plots
│ │ │ │ ├── Absolute_Errors_Cyclohexane-DMF.pdf
│ │ │ │ ├── Absolute_Errors_Cyclohexane-water.pdf
│ │ │ │ ├── Absolute_Errors_Ethyl acetate-water.pdf
│ │ │ │ ├── Absolute_Errors_Heptane-water.pdf
│ │ │ │ ├── Absolute_Errors_MEK-water.pdf
│ │ │ │ ├── Absolute_Errors_Octanol-water.pdf
│ │ │ │ ├── Absolute_Errors_TBME-water.pdf
│ │ │ │ ├── MA_Error_plots
│ │ │ │ ├── mae_Cyclohexane-DMF.pdf
│ │ │ │ ├── mae_Cyclohexane-water.pdf
│ │ │ │ ├── mae_Ethyl acetate-water.pdf
│ │ │ │ ├── mae_Heptane-water.pdf
│ │ │ │ ├── mae_MEK-water.pdf
│ │ │ │ ├── mae_Octanol-water.pdf
│ │ │ │ └── mae_TBME-water.pdf
│ │ │ │ ├── Mean_Error_plots
│ │ │ │ ├── Mean_error_Cyclohexane-DMF.pdf
│ │ │ │ ├── Mean_error_Cyclohexane-water.pdf
│ │ │ │ ├── Mean_error_Ethyl acetate-water.pdf
│ │ │ │ ├── Mean_error_Heptane-water.pdf
│ │ │ │ ├── Mean_error_MEK-water.pdf
│ │ │ │ ├── Mean_error_Octanol-water.pdf
│ │ │ │ └── Mean_error_TBME-water.pdf
│ │ │ │ ├── README.md
│ │ │ │ ├── RMS_Error_plots
│ │ │ │ ├── rmse_Cyclohexane-DMF.pdf
│ │ │ │ ├── rmse_Cyclohexane-water.pdf
│ │ │ │ ├── rmse_Ethyl acetate-water.pdf
│ │ │ │ ├── rmse_Heptane-water.pdf
│ │ │ │ ├── rmse_MEK-water.pdf
│ │ │ │ ├── rmse_Octanol-water.pdf
│ │ │ │ └── rmse_TBME-water.pdf
│ │ │ │ └── error_stats_all_by_sols.csv
│ │ ├── Performance_stats_by_submission
│ │ │ ├── Corr_plots
│ │ │ │ ├── corr_stats_all_combos.csv
│ │ │ │ ├── logD-3DS-1_Corr_plot.pdf
│ │ │ │ ├── logD-ECRISM-1_Corr_plot.pdf
│ │ │ │ ├── logD-ECRISM-2_Corr_plot.pdf
│ │ │ │ ├── logD-ECRISM-3_Corr_plot.pdf
│ │ │ │ ├── logD-davyguan-1_Corr_plot.pdf
│ │ │ │ ├── logD_OllierTranPaluch_LSER_exp_Corr_plot.pdf
│ │ │ │ ├── logD_OllierTranPaluch_UFZ_LSER_exp_Corr_plot.pdf
│ │ │ │ ├── logD_SAMPL8_ShuzheWang_ranked_Corr_plot.pdf
│ │ │ │ ├── logD_SAMPL8_ShuzheWang_unranked1_Corr_plot.pdf
│ │ │ │ ├── logD_SAMPL8_ShuzheWang_unranked2_Corr_plot.pdf
│ │ │ │ ├── logD_SAMPL8_ShuzheWang_unranked3_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_2_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_3_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_2_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_3_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_exp_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_extra_2_Corr_plot.pdf
│ │ │ │ ├── logD_SabatinoRodriguezPaluch_uESE_extra_3_Corr_plot.pdf
│ │ │ │ └── logD_SabatinoRodriguezPaluch_uESE_extra_Corr_plot.pdf
│ │ │ ├── Error_plots
│ │ │ │ ├── Absolute_Errors_all_combo_by_method.pdf
│ │ │ │ └── Absolute_error_all_combo_by_solvent_combo.pdf
│ │ │ └── README.md
│ │ ├── README.md
│ │ ├── logD_all_combos_dataset.csv
│ │ └── logD_dataset.csv
│ ├── analysis_logD.py
│ ├── analysis_ranked
│ │ ├── Performance_stats_by_solvent_combo
│ │ │ └── Error_plots
│ │ │ │ ├── Absolute_Errors_Cyclohexane-DMF.pdf
│ │ │ │ ├── Absolute_Errors_Cyclohexane-water.pdf
│ │ │ │ ├── Absolute_Errors_Ethyl acetate-water.pdf
│ │ │ │ ├── Absolute_Errors_Heptane-water.pdf
│ │ │ │ ├── Absolute_Errors_MEK-water.pdf
│ │ │ │ ├── Absolute_Errors_Octanol-water.pdf
│ │ │ │ ├── Absolute_Errors_TBME-water.pdf
│ │ │ │ ├── MA_Error_plots
│ │ │ │ ├── mae_Cyclohexane-DMF.pdf
│ │ │ │ ├── mae_Cyclohexane-water.pdf
│ │ │ │ ├── mae_Ethyl acetate-water.pdf
│ │ │ │ ├── mae_Heptane-water.pdf
│ │ │ │ ├── mae_MEK-water.pdf
│ │ │ │ ├── mae_Octanol-water.pdf
│ │ │ │ └── mae_TBME-water.pdf
│ │ │ │ ├── Mean_Error_plots
│ │ │ │ ├── Mean_error_Cyclohexane-DMF.pdf
│ │ │ │ ├── Mean_error_Cyclohexane-water.pdf
│ │ │ │ ├── Mean_error_Ethyl acetate-water.pdf
│ │ │ │ ├── Mean_error_Heptane-water.pdf
│ │ │ │ ├── Mean_error_MEK-water.pdf
│ │ │ │ ├── Mean_error_Octanol-water.pdf
│ │ │ │ └── Mean_error_TBME-water.pdf
│ │ │ │ ├── README.md
│ │ │ │ ├── RMS_Error_plots
│ │ │ │ ├── rmse_Cyclohexane-DMF.pdf
│ │ │ │ ├── rmse_Cyclohexane-water.pdf
│ │ │ │ ├── rmse_Ethyl acetate-water.pdf
│ │ │ │ ├── rmse_Heptane-water.pdf
│ │ │ │ ├── rmse_MEK-water.pdf
│ │ │ │ ├── rmse_Octanol-water.pdf
│ │ │ │ └── rmse_TBME-water.pdf
│ │ │ │ └── error_stats_all_by_sols.csv
│ │ ├── Performance_stats_by_submission
│ │ │ ├── Corr_plots
│ │ │ │ ├── corr_stats_all_combos.csv
│ │ │ │ ├── logD-3DS-1_Corr_plot.pdf
│ │ │ │ ├── logD-ECRISM-1_Corr_plot.pdf
│ │ │ │ ├── logD-davyguan-1_Corr_plot.pdf
│ │ │ │ ├── logD_SAMPL8_ShuzheWang_ranked_Corr_plot.pdf
│ │ │ │ └── logD_SabatinoRodriguezPaluch_uESE_extra_Corr_plot.pdf
│ │ │ ├── Error_plots
│ │ │ │ ├── Absolute_Errors_all_combo_by_method.pdf
│ │ │ │ └── Absolute_error_all_combo_by_solvent_combo.pdf
│ │ │ └── README.md
│ │ ├── README.md
│ │ ├── logD_all_combos_dataset.csv
│ │ └── logD_dataset.csv
│ ├── functions_analysis_logD.py
│ └── get_usermap.py
├── example_submission_file
│ ├── logD-example-submission.csv
│ └── logD_test.csv
├── logD_challenge_instructions.md
└── submission_template_file
│ └── logD_prediction_template.csv
├── microstates
├── README.md
├── SAMPL8-1.mol2
├── SAMPL8-1.pdb
├── SAMPL8-1.sdf
├── SAMPL8-10.mol2
├── SAMPL8-10.pdb
├── SAMPL8-10.sdf
├── SAMPL8-10_micro000.mol2
├── SAMPL8-10_micro000.pdb
├── SAMPL8-10_micro000.sdf
├── SAMPL8-10_micro001.mol2
├── SAMPL8-10_micro001.pdb
├── SAMPL8-10_micro001.sdf
├── SAMPL8-10_microstates.csv
├── SAMPL8-11.mol2
├── SAMPL8-11.pdb
├── SAMPL8-11.sdf
├── SAMPL8-11_micro000.mol2
├── SAMPL8-11_micro000.pdb
├── SAMPL8-11_micro000.sdf
├── SAMPL8-11_micro001.mol2
├── SAMPL8-11_micro001.pdb
├── SAMPL8-11_micro001.sdf
├── SAMPL8-11_micro002.mol2
├── SAMPL8-11_micro002.pdb
├── SAMPL8-11_micro002.sdf
├── SAMPL8-11_micro003.mol2
├── SAMPL8-11_micro003.pdb
├── SAMPL8-11_micro003.sdf
├── SAMPL8-11_micro004.mol2
├── SAMPL8-11_micro004.pdb
├── SAMPL8-11_micro004.sdf
├── SAMPL8-11_micro005.mol2
├── SAMPL8-11_micro005.pdb
├── SAMPL8-11_micro005.sdf
├── SAMPL8-11_microstates.csv
├── SAMPL8-12.mol2
├── SAMPL8-12.pdb
├── SAMPL8-12.sdf
├── SAMPL8-12_micro000.mol2
├── SAMPL8-12_micro000.pdb
├── SAMPL8-12_micro000.sdf
├── SAMPL8-12_micro001.mol2
├── SAMPL8-12_micro001.pdb
├── SAMPL8-12_micro001.sdf
├── SAMPL8-12_micro002.mol2
├── SAMPL8-12_micro002.pdb
├── SAMPL8-12_micro002.sdf
├── SAMPL8-12_micro003.mol2
├── SAMPL8-12_micro003.pdb
├── SAMPL8-12_micro003.sdf
├── SAMPL8-12_microstates.csv
├── SAMPL8-13.mol2
├── SAMPL8-13.pdb
├── SAMPL8-13.sdf
├── SAMPL8-13_micro000.mol2
├── SAMPL8-13_micro000.pdb
├── SAMPL8-13_micro000.sdf
├── SAMPL8-13_micro001.mol2
├── SAMPL8-13_micro001.pdb
├── SAMPL8-13_micro001.sdf
├── SAMPL8-13_micro002.mol2
├── SAMPL8-13_micro002.pdb
├── SAMPL8-13_micro002.sdf
├── SAMPL8-13_microstates.csv
├── SAMPL8-14.mol2
├── SAMPL8-14.pdb
├── SAMPL8-14.sdf
├── SAMPL8-14_micro000.mol2
├── SAMPL8-14_micro000.pdb
├── SAMPL8-14_micro000.sdf
├── SAMPL8-14_micro001.mol2
├── SAMPL8-14_micro001.pdb
├── SAMPL8-14_micro001.sdf
├── SAMPL8-14_micro002.mol2
├── SAMPL8-14_micro002.pdb
├── SAMPL8-14_micro002.sdf
├── SAMPL8-14_micro003.mol2
├── SAMPL8-14_micro003.pdb
├── SAMPL8-14_micro003.sdf
├── SAMPL8-14_micro004.mol2
├── SAMPL8-14_micro004.pdb
├── SAMPL8-14_micro004.sdf
├── SAMPL8-14_micro005.mol2
├── SAMPL8-14_micro005.pdb
├── SAMPL8-14_micro005.sdf
├── SAMPL8-14_micro006.mol2
├── SAMPL8-14_micro006.pdb
├── SAMPL8-14_micro006.sdf
├── SAMPL8-14_micro007.mol2
├── SAMPL8-14_micro007.pdb
├── SAMPL8-14_micro007.sdf
├── SAMPL8-14_micro008.mol2
├── SAMPL8-14_micro008.pdb
├── SAMPL8-14_micro008.sdf
├── SAMPL8-14_micro010.mol2
├── SAMPL8-14_micro010.pdb
├── SAMPL8-14_micro010.sdf
├── SAMPL8-14_micro011.mol2
├── SAMPL8-14_micro011.pdb
├── SAMPL8-14_micro011.sdf
├── SAMPL8-14_micro012.mol2
├── SAMPL8-14_micro012.pdb
├── SAMPL8-14_micro012.sdf
├── SAMPL8-14_micro013.mol2
├── SAMPL8-14_micro013.pdb
├── SAMPL8-14_micro013.sdf
├── SAMPL8-14_micro014.mol2
├── SAMPL8-14_micro014.pdb
├── SAMPL8-14_micro014.sdf
├── SAMPL8-14_micro015.mol2
├── SAMPL8-14_micro015.pdb
├── SAMPL8-14_micro015.sdf
├── SAMPL8-14_micro016.mol2
├── SAMPL8-14_micro016.pdb
├── SAMPL8-14_micro016.sdf
├── SAMPL8-14_micro017.mol2
├── SAMPL8-14_micro017.pdb
├── SAMPL8-14_micro017.sdf
├── SAMPL8-14_micro018.mol2
├── SAMPL8-14_micro018.pdb
├── SAMPL8-14_micro018.sdf
├── SAMPL8-14_micro019.mol2
├── SAMPL8-14_micro019.pdb
├── SAMPL8-14_micro019.sdf
├── SAMPL8-14_micro020.mol2
├── SAMPL8-14_micro020.pdb
├── SAMPL8-14_micro020.sdf
├── SAMPL8-14_micro021.mol2
├── SAMPL8-14_micro021.pdb
├── SAMPL8-14_micro021.sdf
├── SAMPL8-14_micro022.mol2
├── SAMPL8-14_micro022.pdb
├── SAMPL8-14_micro022.sdf
├── SAMPL8-14_micro023.mol2
├── SAMPL8-14_micro023.pdb
├── SAMPL8-14_micro023.sdf
├── SAMPL8-14_micro024.mol2
├── SAMPL8-14_micro024.pdb
├── SAMPL8-14_micro024.sdf
├── SAMPL8-14_micro025.mol2
├── SAMPL8-14_micro025.pdb
├── SAMPL8-14_micro025.sdf
├── SAMPL8-14_micro026.mol2
├── SAMPL8-14_micro026.pdb
├── SAMPL8-14_micro026.sdf
├── SAMPL8-14_micro027.mol2
├── SAMPL8-14_micro027.pdb
├── SAMPL8-14_micro027.sdf
├── SAMPL8-14_micro028.mol2
├── SAMPL8-14_micro028.pdb
├── SAMPL8-14_micro028.sdf
├── SAMPL8-14_micro029.mol2
├── SAMPL8-14_micro029.pdb
├── SAMPL8-14_micro029.sdf
├── SAMPL8-14_micro030.mol2
├── SAMPL8-14_micro030.pdb
├── SAMPL8-14_micro030.sdf
├── SAMPL8-14_micro031.mol2
├── SAMPL8-14_micro031.pdb
├── SAMPL8-14_micro031.sdf
├── SAMPL8-14_micro032.mol2
├── SAMPL8-14_micro032.pdb
├── SAMPL8-14_micro032.sdf
├── SAMPL8-14_micro033.mol2
├── SAMPL8-14_micro033.pdb
├── SAMPL8-14_micro033.sdf
├── SAMPL8-14_micro034.mol2
├── SAMPL8-14_micro034.pdb
├── SAMPL8-14_micro034.sdf
├── SAMPL8-14_micro09.mol2
├── SAMPL8-14_micro09.pdb
├── SAMPL8-14_micro09.sdf
├── SAMPL8-14_microstates.csv
├── SAMPL8-15.mol2
├── SAMPL8-15.pdb
├── SAMPL8-15.sdf
├── SAMPL8-15_micro000.mol2
├── SAMPL8-15_micro000.pdb
├── SAMPL8-15_micro000.sdf
├── SAMPL8-15_micro001.mol2
├── SAMPL8-15_micro001.pdb
├── SAMPL8-15_micro001.sdf
├── SAMPL8-15_micro002.mol2
├── SAMPL8-15_micro002.pdb
├── SAMPL8-15_micro002.sdf
├── SAMPL8-15_micro003.mol2
├── SAMPL8-15_micro003.pdb
├── SAMPL8-15_micro003.sdf
├── SAMPL8-15_micro004.mol2
├── SAMPL8-15_micro004.pdb
├── SAMPL8-15_micro004.sdf
├── SAMPL8-15_microstates.csv
├── SAMPL8-16.mol2
├── SAMPL8-16.pdb
├── SAMPL8-16.sdf
├── SAMPL8-16_micro000.mol2
├── SAMPL8-16_micro000.pdb
├── SAMPL8-16_micro000.sdf
├── SAMPL8-16_micro001.mol2
├── SAMPL8-16_micro001.pdb
├── SAMPL8-16_micro001.sdf
├── SAMPL8-16_micro002.mol2
├── SAMPL8-16_micro002.pdb
├── SAMPL8-16_micro002.sdf
├── SAMPL8-16_micro003.mol2
├── SAMPL8-16_micro003.pdb
├── SAMPL8-16_micro003.sdf
├── SAMPL8-16_micro004.mol2
├── SAMPL8-16_micro004.pdb
├── SAMPL8-16_micro004.sdf
├── SAMPL8-16_micro005.mol2
├── SAMPL8-16_micro005.pdb
├── SAMPL8-16_micro005.sdf
├── SAMPL8-16_micro006.mol2
├── SAMPL8-16_micro006.pdb
├── SAMPL8-16_micro006.sdf
├── SAMPL8-16_micro007.mol2
├── SAMPL8-16_micro007.pdb
├── SAMPL8-16_micro007.sdf
├── SAMPL8-16_micro008.mol2
├── SAMPL8-16_micro008.pdb
├── SAMPL8-16_micro008.sdf
├── SAMPL8-16_micro009.mol2
├── SAMPL8-16_micro009.pdb
├── SAMPL8-16_micro009.sdf
├── SAMPL8-16_micro010.mol2
├── SAMPL8-16_micro010.pdb
├── SAMPL8-16_micro010.sdf
├── SAMPL8-16_micro011.mol2
├── SAMPL8-16_micro011.pdb
├── SAMPL8-16_micro011.sdf
├── SAMPL8-16_microstates.csv
├── SAMPL8-17.mol2
├── SAMPL8-17.pdb
├── SAMPL8-17.sdf
├── SAMPL8-17_micro000.mol2
├── SAMPL8-17_micro000.pdb
├── SAMPL8-17_micro000.sdf
├── SAMPL8-17_micro001.mol2
├── SAMPL8-17_micro001.pdb
├── SAMPL8-17_micro001.sdf
├── SAMPL8-17_micro002.mol2
├── SAMPL8-17_micro002.pdb
├── SAMPL8-17_micro002.sdf
├── SAMPL8-17_micro003.mol2
├── SAMPL8-17_micro003.pdb
├── SAMPL8-17_micro003.sdf
├── SAMPL8-17_micro004.mol2
├── SAMPL8-17_micro004.pdb
├── SAMPL8-17_micro004.sdf
├── SAMPL8-17_micro005.mol2
├── SAMPL8-17_micro005.pdb
├── SAMPL8-17_micro005.sdf
├── SAMPL8-17_microstates.csv
├── SAMPL8-18.mol2
├── SAMPL8-18.pdb
├── SAMPL8-18.sdf
├── SAMPL8-18_micro000.mol2
├── SAMPL8-18_micro000.pdb
├── SAMPL8-18_micro000.sdf
├── SAMPL8-18_micro001.mol2
├── SAMPL8-18_micro001.pdb
├── SAMPL8-18_micro001.sdf
├── SAMPL8-18_micro002.mol2
├── SAMPL8-18_micro002.pdb
├── SAMPL8-18_micro002.sdf
├── SAMPL8-18_micro003.mol2
├── SAMPL8-18_micro003.pdb
├── SAMPL8-18_micro003.sdf
├── SAMPL8-18_micro004.mol2
├── SAMPL8-18_micro004.pdb
├── SAMPL8-18_micro004.sdf
├── SAMPL8-18_micro005.mol2
├── SAMPL8-18_micro005.pdb
├── SAMPL8-18_micro005.sdf
├── SAMPL8-18_microstates.csv
├── SAMPL8-19.mol2
├── SAMPL8-19.pdb
├── SAMPL8-19.sdf
├── SAMPL8-19_micro000.mol2
├── SAMPL8-19_micro000.pdb
├── SAMPL8-19_micro000.sdf
├── SAMPL8-19_micro001.mol2
├── SAMPL8-19_micro001.pdb
├── SAMPL8-19_micro001.sdf
├── SAMPL8-19_micro002.mol2
├── SAMPL8-19_micro002.pdb
├── SAMPL8-19_micro002.sdf
├── SAMPL8-19_micro003.mol2
├── SAMPL8-19_micro003.pdb
├── SAMPL8-19_micro003.sdf
├── SAMPL8-19_micro004.mol2
├── SAMPL8-19_micro004.pdb
├── SAMPL8-19_micro004.sdf
├── SAMPL8-19_micro005.mol2
├── SAMPL8-19_micro005.pdb
├── SAMPL8-19_micro005.sdf
├── SAMPL8-19_micro006.mol2
├── SAMPL8-19_micro006.pdb
├── SAMPL8-19_micro006.sdf
├── SAMPL8-19_micro007.mol2
├── SAMPL8-19_micro007.pdb
├── SAMPL8-19_micro007.sdf
├── SAMPL8-19_micro008.mol2
├── SAMPL8-19_micro008.pdb
├── SAMPL8-19_micro008.sdf
├── SAMPL8-19_micro009.mol2
├── SAMPL8-19_micro009.pdb
├── SAMPL8-19_micro009.sdf
├── SAMPL8-19_micro010.mol2
├── SAMPL8-19_micro010.pdb
├── SAMPL8-19_micro010.sdf
├── SAMPL8-19_micro011.mol2
├── SAMPL8-19_micro011.pdb
├── SAMPL8-19_micro011.sdf
├── SAMPL8-19_micro012.mol2
├── SAMPL8-19_micro012.pdb
├── SAMPL8-19_micro012.sdf
├── SAMPL8-19_micro013.mol2
├── SAMPL8-19_micro013.pdb
├── SAMPL8-19_micro013.sdf
├── SAMPL8-19_micro014.mol2
├── SAMPL8-19_micro014.pdb
├── SAMPL8-19_micro014.sdf
├── SAMPL8-19_micro015.mol2
├── SAMPL8-19_micro015.pdb
├── SAMPL8-19_micro015.sdf
├── SAMPL8-19_micro016.mol2
├── SAMPL8-19_micro016.pdb
├── SAMPL8-19_micro016.sdf
├── SAMPL8-19_micro017.mol2
├── SAMPL8-19_micro017.pdb
├── SAMPL8-19_micro017.sdf
├── SAMPL8-19_micro018.mol2
├── SAMPL8-19_micro018.pdb
├── SAMPL8-19_micro018.sdf
├── SAMPL8-19_micro019.mol2
├── SAMPL8-19_micro019.pdb
├── SAMPL8-19_micro019.sdf
├── SAMPL8-19_micro020.mol2
├── SAMPL8-19_micro020.pdb
├── SAMPL8-19_micro020.sdf
├── SAMPL8-19_micro021.mol2
├── SAMPL8-19_micro021.pdb
├── SAMPL8-19_micro021.sdf
├── SAMPL8-19_micro022.mol2
├── SAMPL8-19_micro022.pdb
├── SAMPL8-19_micro022.sdf
├── SAMPL8-19_micro023.mol2
├── SAMPL8-19_micro023.pdb
├── SAMPL8-19_micro023.sdf
├── SAMPL8-19_micro024.mol2
├── SAMPL8-19_micro024.pdb
├── SAMPL8-19_micro024.sdf
├── SAMPL8-19_micro025.mol2
├── SAMPL8-19_micro025.pdb
├── SAMPL8-19_micro025.sdf
├── SAMPL8-19_microstates.csv
├── SAMPL8-1_micro000.mol2
├── SAMPL8-1_micro000.pdb
├── SAMPL8-1_micro000.sdf
├── SAMPL8-1_micro001.mol2
├── SAMPL8-1_micro001.pdb
├── SAMPL8-1_micro001.sdf
├── SAMPL8-1_micro002.mol2
├── SAMPL8-1_micro002.pdb
├── SAMPL8-1_micro002.sdf
├── SAMPL8-1_micro003.mol2
├── SAMPL8-1_micro003.pdb
├── SAMPL8-1_micro003.sdf
├── SAMPL8-1_micro004.mol2
├── SAMPL8-1_micro004.pdb
├── SAMPL8-1_micro004.sdf
├── SAMPL8-1_micro005.mol2
├── SAMPL8-1_micro005.pdb
├── SAMPL8-1_micro005.sdf
├── SAMPL8-1_micro006.mol2
├── SAMPL8-1_micro006.pdb
├── SAMPL8-1_micro006.sdf
├── SAMPL8-1_micro007.mol2
├── SAMPL8-1_micro007.pdb
├── SAMPL8-1_micro007.sdf
├── SAMPL8-1_micro008.mol2
├── SAMPL8-1_micro008.pdb
├── SAMPL8-1_micro008.sdf
├── SAMPL8-1_micro009.mol2
├── SAMPL8-1_micro009.pdb
├── SAMPL8-1_micro009.sdf
├── SAMPL8-1_micro010.mol2
├── SAMPL8-1_micro010.pdb
├── SAMPL8-1_micro010.sdf
├── SAMPL8-1_microstates.csv
├── SAMPL8-2.mol2
├── SAMPL8-2.pdb
├── SAMPL8-2.sdf
├── SAMPL8-20.mol2
├── SAMPL8-20.pdb
├── SAMPL8-20.sdf
├── SAMPL8-20_micro000.mol2
├── SAMPL8-20_micro000.pdb
├── SAMPL8-20_micro000.sdf
├── SAMPL8-20_micro001.mol2
├── SAMPL8-20_micro001.pdb
├── SAMPL8-20_micro001.sdf
├── SAMPL8-20_micro002.mol2
├── SAMPL8-20_micro002.pdb
├── SAMPL8-20_micro002.sdf
├── SAMPL8-20_micro003.mol2
├── SAMPL8-20_micro003.pdb
├── SAMPL8-20_micro003.sdf
├── SAMPL8-20_micro004.mol2
├── SAMPL8-20_micro004.pdb
├── SAMPL8-20_micro004.sdf
├── SAMPL8-20_micro005.mol2
├── SAMPL8-20_micro005.pdb
├── SAMPL8-20_micro005.sdf
├── SAMPL8-20_micro006.mol2
├── SAMPL8-20_micro006.pdb
├── SAMPL8-20_micro006.sdf
├── SAMPL8-20_micro007.mol2
├── SAMPL8-20_micro007.pdb
├── SAMPL8-20_micro007.sdf
├── SAMPL8-20_micro008.mol2
├── SAMPL8-20_micro008.pdb
├── SAMPL8-20_micro008.sdf
├── SAMPL8-20_micro009.mol2
├── SAMPL8-20_micro009.pdb
├── SAMPL8-20_micro009.sdf
├── SAMPL8-20_micro010.mol2
├── SAMPL8-20_micro010.pdb
├── SAMPL8-20_micro010.sdf
├── SAMPL8-20_micro011.mol2
├── SAMPL8-20_micro011.pdb
├── SAMPL8-20_micro011.sdf
├── SAMPL8-20_micro012.mol2
├── SAMPL8-20_micro012.pdb
├── SAMPL8-20_micro012.sdf
├── SAMPL8-20_micro013.mol2
├── SAMPL8-20_micro013.pdb
├── SAMPL8-20_micro013.sdf
├── SAMPL8-20_micro014.mol2
├── SAMPL8-20_micro014.pdb
├── SAMPL8-20_micro014.sdf
├── SAMPL8-20_micro015.mol2
├── SAMPL8-20_micro015.pdb
├── SAMPL8-20_micro015.sdf
├── SAMPL8-20_micro016.mol2
├── SAMPL8-20_micro016.pdb
├── SAMPL8-20_micro016.sdf
├── SAMPL8-20_micro017.mol2
├── SAMPL8-20_micro017.pdb
├── SAMPL8-20_micro017.sdf
├── SAMPL8-20_micro018.mol2
├── SAMPL8-20_micro018.pdb
├── SAMPL8-20_micro018.sdf
├── SAMPL8-20_micro019.mol2
├── SAMPL8-20_micro019.pdb
├── SAMPL8-20_micro019.sdf
├── SAMPL8-20_micro020.mol2
├── SAMPL8-20_micro020.pdb
├── SAMPL8-20_micro020.sdf
├── SAMPL8-20_micro021.mol2
├── SAMPL8-20_micro021.pdb
├── SAMPL8-20_micro021.sdf
├── SAMPL8-20_micro022.mol2
├── SAMPL8-20_micro022.pdb
├── SAMPL8-20_micro022.sdf
├── SAMPL8-20_micro023.mol2
├── SAMPL8-20_micro023.pdb
├── SAMPL8-20_micro023.sdf
├── SAMPL8-20_micro024.mol2
├── SAMPL8-20_micro024.pdb
├── SAMPL8-20_micro024.sdf
├── SAMPL8-20_micro025.mol2
├── SAMPL8-20_micro025.pdb
├── SAMPL8-20_micro025.sdf
├── SAMPL8-20_micro026.mol2
├── SAMPL8-20_micro026.pdb
├── SAMPL8-20_micro026.sdf
├── SAMPL8-20_micro027.mol2
├── SAMPL8-20_micro027.pdb
├── SAMPL8-20_micro027.sdf
├── SAMPL8-20_micro028.mol2
├── SAMPL8-20_micro028.pdb
├── SAMPL8-20_micro028.sdf
├── SAMPL8-20_microstates.csv
├── SAMPL8-21.mol2
├── SAMPL8-21.pdb
├── SAMPL8-21.sdf
├── SAMPL8-21_micro000.mol2
├── SAMPL8-21_micro000.pdb
├── SAMPL8-21_micro000.sdf
├── SAMPL8-21_micro001.mol2
├── SAMPL8-21_micro001.pdb
├── SAMPL8-21_micro001.sdf
├── SAMPL8-21_micro002.mol2
├── SAMPL8-21_micro002.pdb
├── SAMPL8-21_micro002.sdf
├── SAMPL8-21_micro003.mol2
├── SAMPL8-21_micro003.pdb
├── SAMPL8-21_micro003.sdf
├── SAMPL8-21_micro004.mol2
├── SAMPL8-21_micro004.pdb
├── SAMPL8-21_micro004.sdf
├── SAMPL8-21_micro005.mol2
├── SAMPL8-21_micro005.pdb
├── SAMPL8-21_micro005.sdf
├── SAMPL8-21_micro006.mol2
├── SAMPL8-21_micro006.pdb
├── SAMPL8-21_micro006.sdf
├── SAMPL8-21_micro007.mol2
├── SAMPL8-21_micro007.pdb
├── SAMPL8-21_micro007.sdf
├── SAMPL8-21_micro008.mol2
├── SAMPL8-21_micro008.pdb
├── SAMPL8-21_micro008.sdf
├── SAMPL8-21_micro009.mol2
├── SAMPL8-21_micro009.pdb
├── SAMPL8-21_micro009.sdf
├── SAMPL8-21_micro010.mol2
├── SAMPL8-21_micro010.pdb
├── SAMPL8-21_micro010.sdf
├── SAMPL8-21_micro011.mol2
├── SAMPL8-21_micro011.pdb
├── SAMPL8-21_micro011.sdf
├── SAMPL8-21_micro012.mol2
├── SAMPL8-21_micro012.pdb
├── SAMPL8-21_micro012.sdf
├── SAMPL8-21_micro013.mol2
├── SAMPL8-21_micro013.pdb
├── SAMPL8-21_micro013.sdf
├── SAMPL8-21_micro014.mol2
├── SAMPL8-21_micro014.pdb
├── SAMPL8-21_micro014.sdf
├── SAMPL8-21_micro015.mol2
├── SAMPL8-21_micro015.pdb
├── SAMPL8-21_micro015.sdf
├── SAMPL8-21_micro016.mol2
├── SAMPL8-21_micro016.pdb
├── SAMPL8-21_micro016.sdf
├── SAMPL8-21_micro017.mol2
├── SAMPL8-21_micro017.pdb
├── SAMPL8-21_micro017.sdf
├── SAMPL8-21_micro018.mol2
├── SAMPL8-21_micro018.pdb
├── SAMPL8-21_micro018.sdf
├── SAMPL8-21_micro019.mol2
├── SAMPL8-21_micro019.pdb
├── SAMPL8-21_micro019.sdf
├── SAMPL8-21_micro020.mol2
├── SAMPL8-21_micro020.pdb
├── SAMPL8-21_micro020.sdf
├── SAMPL8-21_micro021.mol2
├── SAMPL8-21_micro021.pdb
├── SAMPL8-21_micro021.sdf
├── SAMPL8-21_micro022.mol2
├── SAMPL8-21_micro022.pdb
├── SAMPL8-21_micro022.sdf
├── SAMPL8-21_micro023.mol2
├── SAMPL8-21_micro023.pdb
├── SAMPL8-21_micro023.sdf
├── SAMPL8-21_micro024.mol2
├── SAMPL8-21_micro024.pdb
├── SAMPL8-21_micro024.sdf
├── SAMPL8-21_micro025.mol2
├── SAMPL8-21_micro025.pdb
├── SAMPL8-21_micro025.sdf
├── SAMPL8-21_micro026.mol2
├── SAMPL8-21_micro026.pdb
├── SAMPL8-21_micro026.sdf
├── SAMPL8-21_micro027.mol2
├── SAMPL8-21_micro027.pdb
├── SAMPL8-21_micro027.sdf
├── SAMPL8-21_micro028.mol2
├── SAMPL8-21_micro028.pdb
├── SAMPL8-21_micro028.sdf
├── SAMPL8-21_micro029.mol2
├── SAMPL8-21_micro029.pdb
├── SAMPL8-21_micro029.sdf
├── SAMPL8-21_microstates.csv
├── SAMPL8-22.mol2
├── SAMPL8-22.pdb
├── SAMPL8-22.sdf
├── SAMPL8-22_micro000.mol2
├── SAMPL8-22_micro000.pdb
├── SAMPL8-22_micro000.sdf
├── SAMPL8-22_micro001.mol2
├── SAMPL8-22_micro001.pdb
├── SAMPL8-22_micro001.sdf
├── SAMPL8-22_micro002.mol2
├── SAMPL8-22_micro002.pdb
├── SAMPL8-22_micro002.sdf
├── SAMPL8-22_micro003.mol2
├── SAMPL8-22_micro003.pdb
├── SAMPL8-22_micro003.sdf
├── SAMPL8-22_microstates.csv
├── SAMPL8-23.mol2
├── SAMPL8-23.pdb
├── SAMPL8-23.sdf
├── SAMPL8-23_micro000.mol2
├── SAMPL8-23_micro000.pdb
├── SAMPL8-23_micro000.sdf
├── SAMPL8-23_micro001.mol2
├── SAMPL8-23_micro001.pdb
├── SAMPL8-23_micro001.sdf
├── SAMPL8-23_micro002.mol2
├── SAMPL8-23_micro002.pdb
├── SAMPL8-23_micro002.sdf
├── SAMPL8-23_micro003.mol2
├── SAMPL8-23_micro003.pdb
├── SAMPL8-23_micro003.sdf
├── SAMPL8-23_micro004.mol2
├── SAMPL8-23_micro004.pdb
├── SAMPL8-23_micro004.sdf
├── SAMPL8-23_micro005.mol2
├── SAMPL8-23_micro005.pdb
├── SAMPL8-23_micro005.sdf
├── SAMPL8-23_micro006.mol2
├── SAMPL8-23_micro006.pdb
├── SAMPL8-23_micro006.sdf
├── SAMPL8-23_micro007.mol2
├── SAMPL8-23_micro007.pdb
├── SAMPL8-23_micro007.sdf
├── SAMPL8-23_microstates.csv
├── SAMPL8-2_micro000.mol2
├── SAMPL8-2_micro000.pdb
├── SAMPL8-2_micro000.sdf
├── SAMPL8-2_micro001.mol2
├── SAMPL8-2_micro001.pdb
├── SAMPL8-2_micro001.sdf
├── SAMPL8-2_micro002.mol2
├── SAMPL8-2_micro002.pdb
├── SAMPL8-2_micro002.sdf
├── SAMPL8-2_micro003.mol2
├── SAMPL8-2_micro003.pdb
├── SAMPL8-2_micro003.sdf
├── SAMPL8-2_microstates.csv
├── SAMPL8-3.mol2
├── SAMPL8-3.pdb
├── SAMPL8-3.sdf
├── SAMPL8-3_micro000.mol2
├── SAMPL8-3_micro000.pdb
├── SAMPL8-3_micro000.sdf
├── SAMPL8-3_micro001.mol2
├── SAMPL8-3_micro001.pdb
├── SAMPL8-3_micro001.sdf
├── SAMPL8-3_micro002.mol2
├── SAMPL8-3_micro002.pdb
├── SAMPL8-3_micro002.sdf
├── SAMPL8-3_micro003.mol2
├── SAMPL8-3_micro003.pdb
├── SAMPL8-3_micro003.sdf
├── SAMPL8-3_micro004.mol2
├── SAMPL8-3_micro004.pdb
├── SAMPL8-3_micro004.sdf
├── SAMPL8-3_micro005.mol2
├── SAMPL8-3_micro005.pdb
├── SAMPL8-3_micro005.sdf
├── SAMPL8-3_micro006.mol2
├── SAMPL8-3_micro006.pdb
├── SAMPL8-3_micro006.sdf
├── SAMPL8-3_micro007.mol2
├── SAMPL8-3_micro007.pdb
├── SAMPL8-3_micro007.sdf
├── SAMPL8-3_micro008.mol2
├── SAMPL8-3_micro008.pdb
├── SAMPL8-3_micro008.sdf
├── SAMPL8-3_micro009.mol2
├── SAMPL8-3_micro009.pdb
├── SAMPL8-3_micro009.sdf
├── SAMPL8-3_micro010.mol2
├── SAMPL8-3_micro010.pdb
├── SAMPL8-3_micro010.sdf
├── SAMPL8-3_micro011.mol2
├── SAMPL8-3_micro011.pdb
├── SAMPL8-3_micro011.sdf
├── SAMPL8-3_micro012.mol2
├── SAMPL8-3_micro012.pdb
├── SAMPL8-3_micro012.sdf
├── SAMPL8-3_micro013.mol2
├── SAMPL8-3_micro013.pdb
├── SAMPL8-3_micro013.sdf
├── SAMPL8-3_micro014.mol2
├── SAMPL8-3_micro014.pdb
├── SAMPL8-3_micro014.sdf
├── SAMPL8-3_micro015.mol2
├── SAMPL8-3_micro015.pdb
├── SAMPL8-3_micro015.sdf
├── SAMPL8-3_micro016.mol2
├── SAMPL8-3_micro016.pdb
├── SAMPL8-3_micro016.sdf
├── SAMPL8-3_micro017.mol2
├── SAMPL8-3_micro017.pdb
├── SAMPL8-3_micro017.sdf
├── SAMPL8-3_micro018.mol2
├── SAMPL8-3_micro018.pdb
├── SAMPL8-3_micro018.sdf
├── SAMPL8-3_micro019.mol2
├── SAMPL8-3_micro019.pdb
├── SAMPL8-3_micro019.sdf
├── SAMPL8-3_micro020.mol2
├── SAMPL8-3_micro020.pdb
├── SAMPL8-3_micro020.sdf
├── SAMPL8-3_micro021.mol2
├── SAMPL8-3_micro021.pdb
├── SAMPL8-3_micro021.sdf
├── SAMPL8-3_microstates.csv
├── SAMPL8-4.mol2
├── SAMPL8-4.pdb
├── SAMPL8-4.sdf
├── SAMPL8-4_micro000.mol2
├── SAMPL8-4_micro000.pdb
├── SAMPL8-4_micro000.sdf
├── SAMPL8-4_micro001.mol2
├── SAMPL8-4_micro001.pdb
├── SAMPL8-4_micro001.sdf
├── SAMPL8-4_micro002.mol2
├── SAMPL8-4_micro002.pdb
├── SAMPL8-4_micro002.sdf
├── SAMPL8-4_micro003.mol2
├── SAMPL8-4_micro003.pdb
├── SAMPL8-4_micro003.sdf
├── SAMPL8-4_micro004.mol2
├── SAMPL8-4_micro004.pdb
├── SAMPL8-4_micro004.sdf
├── SAMPL8-4_micro005.mol2
├── SAMPL8-4_micro005.pdb
├── SAMPL8-4_micro005.sdf
├── SAMPL8-4_micro006.mol2
├── SAMPL8-4_micro006.pdb
├── SAMPL8-4_micro006.sdf
├── SAMPL8-4_micro007.mol2
├── SAMPL8-4_micro007.pdb
├── SAMPL8-4_micro007.sdf
├── SAMPL8-4_micro008.mol2
├── SAMPL8-4_micro008.pdb
├── SAMPL8-4_micro008.sdf
├── SAMPL8-4_micro009.mol2
├── SAMPL8-4_micro009.pdb
├── SAMPL8-4_micro009.sdf
├── SAMPL8-4_micro010.mol2
├── SAMPL8-4_micro010.pdb
├── SAMPL8-4_micro010.sdf
├── SAMPL8-4_microstates.csv
├── SAMPL8-5.mol2
├── SAMPL8-5.pdb
├── SAMPL8-5.sdf
├── SAMPL8-5_micro000.mol2
├── SAMPL8-5_micro000.pdb
├── SAMPL8-5_micro000.sdf
├── SAMPL8-5_micro001.mol2
├── SAMPL8-5_micro001.pdb
├── SAMPL8-5_micro001.sdf
├── SAMPL8-5_micro002.mol2
├── SAMPL8-5_micro002.pdb
├── SAMPL8-5_micro002.sdf
├── SAMPL8-5_micro003.mol2
├── SAMPL8-5_micro003.pdb
├── SAMPL8-5_micro003.sdf
├── SAMPL8-5_micro004.mol2
├── SAMPL8-5_micro004.pdb
├── SAMPL8-5_micro004.sdf
├── SAMPL8-5_micro005.mol2
├── SAMPL8-5_micro005.pdb
├── SAMPL8-5_micro005.sdf
├── SAMPL8-5_micro006.mol2
├── SAMPL8-5_micro006.pdb
├── SAMPL8-5_micro006.sdf
├── SAMPL8-5_micro007.mol2
├── SAMPL8-5_micro007.pdb
├── SAMPL8-5_micro007.sdf
├── SAMPL8-5_microstates.csv
├── SAMPL8-6.mol2
├── SAMPL8-6.pdb
├── SAMPL8-6.sdf
├── SAMPL8-6_micro000.mol2
├── SAMPL8-6_micro000.pdb
├── SAMPL8-6_micro000.sdf
├── SAMPL8-6_micro001.mol2
├── SAMPL8-6_micro001.pdb
├── SAMPL8-6_micro001.sdf
├── SAMPL8-6_micro002.mol2
├── SAMPL8-6_micro002.pdb
├── SAMPL8-6_micro002.sdf
├── SAMPL8-6_micro003.mol2
├── SAMPL8-6_micro003.pdb
├── SAMPL8-6_micro003.sdf
├── SAMPL8-6_micro004.mol2
├── SAMPL8-6_micro004.pdb
├── SAMPL8-6_micro004.sdf
├── SAMPL8-6_micro005.mol2
├── SAMPL8-6_micro005.pdb
├── SAMPL8-6_micro005.sdf
├── SAMPL8-6_micro006.mol2
├── SAMPL8-6_micro006.pdb
├── SAMPL8-6_micro006.sdf
├── SAMPL8-6_micro007.mol2
├── SAMPL8-6_micro007.pdb
├── SAMPL8-6_micro007.sdf
├── SAMPL8-6_micro008.mol2
├── SAMPL8-6_micro008.pdb
├── SAMPL8-6_micro008.sdf
├── SAMPL8-6_micro009.mol2
├── SAMPL8-6_micro009.pdb
├── SAMPL8-6_micro009.sdf
├── SAMPL8-6_microstates.csv
├── SAMPL8-7.mol2
├── SAMPL8-7.pdb
├── SAMPL8-7.sdf
├── SAMPL8-7_micro000.mol2
├── SAMPL8-7_micro000.pdb
├── SAMPL8-7_micro000.sdf
├── SAMPL8-7_micro001.mol2
├── SAMPL8-7_micro001.pdb
├── SAMPL8-7_micro001.sdf
├── SAMPL8-7_micro002.mol2
├── SAMPL8-7_micro002.pdb
├── SAMPL8-7_micro002.sdf
├── SAMPL8-7_micro003.mol2
├── SAMPL8-7_micro003.pdb
├── SAMPL8-7_micro003.sdf
├── SAMPL8-7_micro004.mol2
├── SAMPL8-7_micro004.pdb
├── SAMPL8-7_micro004.sdf
├── SAMPL8-7_microstates.csv
├── SAMPL8-8.mol2
├── SAMPL8-8.pdb
├── SAMPL8-8.sdf
├── SAMPL8-8_micro000.mol2
├── SAMPL8-8_micro000.pdb
├── SAMPL8-8_micro000.sdf
├── SAMPL8-8_micro001.mol2
├── SAMPL8-8_micro001.pdb
├── SAMPL8-8_micro001.sdf
├── SAMPL8-8_micro002.mol2
├── SAMPL8-8_micro002.pdb
├── SAMPL8-8_micro002.sdf
├── SAMPL8-8_microstates.csv
├── SAMPL8-9.mol2
├── SAMPL8-9.pdb
├── SAMPL8-9.sdf
├── SAMPL8-9_micro000.mol2
├── SAMPL8-9_micro000.pdb
├── SAMPL8-9_micro000.sdf
├── SAMPL8-9_micro001.mol2
├── SAMPL8-9_micro001.pdb
├── SAMPL8-9_micro001.sdf
├── SAMPL8-9_micro002.mol2
├── SAMPL8-9_micro002.pdb
├── SAMPL8-9_micro002.sdf
├── SAMPL8-9_micro003.mol2
├── SAMPL8-9_micro003.pdb
├── SAMPL8-9_micro003.sdf
├── SAMPL8-9_micro004.mol2
├── SAMPL8-9_micro004.pdb
├── SAMPL8-9_micro004.sdf
├── SAMPL8-9_microstates.csv
├── SAMPL8_molecule_ID_and_SMILES.csv
├── dassault_microstates
│ ├── SAMPL8-10_micro000_c0.mol2
│ ├── SAMPL8-10_micro001_c0.mol2
│ ├── SAMPL8-11_micro000_c0.mol2
│ ├── SAMPL8-11_micro001_c0.mol2
│ ├── SAMPL8-11_micro002_c0.mol2
│ ├── SAMPL8-11_micro003_c0.mol2
│ ├── SAMPL8-11_micro004_c0.mol2
│ ├── SAMPL8-11_micro005_c0.mol2
│ ├── SAMPL8-12_extra001_c0.mol2
│ ├── SAMPL8-12_extra002_c0.mol2
│ ├── SAMPL8-12_extra003_c0.mol2
│ ├── SAMPL8-12_extra004_c0.mol2
│ ├── SAMPL8-12_extra005_c0.mol2
│ ├── SAMPL8-12_extra007_c0.mol2
│ ├── SAMPL8-12_extra008_c0.mol2
│ ├── SAMPL8-12_extra009_c0.mol2
│ ├── SAMPL8-12_micro000_c0.mol2
│ ├── SAMPL8-12_micro001_c0.mol2
│ ├── SAMPL8-12_micro002_c0.mol2
│ ├── SAMPL8-12_micro003_c0.mol2
│ ├── SAMPL8-13_extra001_c0.mol2
│ ├── SAMPL8-13_micro000_c0.mol2
│ ├── SAMPL8-13_micro001_c0.mol2
│ ├── SAMPL8-13_micro002_c0.mol2
│ ├── SAMPL8-14_extra001_c0.mol2
│ ├── SAMPL8-14_extra002_c0.mol2
│ ├── SAMPL8-14_extra003_c0.mol2
│ ├── SAMPL8-14_extra004_c0.mol2
│ ├── SAMPL8-14_extra005_c0.mol2
│ ├── SAMPL8-14_extra006_c0.mol2
│ ├── SAMPL8-14_extra007_c0.mol2
│ ├── SAMPL8-14_extra008_c0.mol2
│ ├── SAMPL8-14_extra009_c0.mol2
│ ├── SAMPL8-14_extra010_c0.mol2
│ ├── SAMPL8-14_micro000_c0.mol2
│ ├── SAMPL8-14_micro001_c0.mol2
│ ├── SAMPL8-14_micro002_c0.mol2
│ ├── SAMPL8-14_micro003_c0.mol2
│ ├── SAMPL8-14_micro004_c0.mol2
│ ├── SAMPL8-14_micro005_c0.mol2
│ ├── SAMPL8-14_micro007_c0.mol2
│ ├── SAMPL8-14_micro008_c0.mol2
│ ├── SAMPL8-14_micro010_c0.mol2
│ ├── SAMPL8-14_micro013_c0.mol2
│ ├── SAMPL8-14_micro017_c0.mol2
│ ├── SAMPL8-14_micro018_c0.mol2
│ ├── SAMPL8-14_micro020_c0.mol2
│ ├── SAMPL8-14_micro021_c0.mol2
│ ├── SAMPL8-14_micro022_c0.mol2
│ ├── SAMPL8-14_micro024_c0.mol2
│ ├── SAMPL8-14_micro027_c0.mol2
│ ├── SAMPL8-14_micro028_c0.mol2
│ ├── SAMPL8-14_micro029_c0.mol2
│ ├── SAMPL8-14_micro032_c0.mol2
│ ├── SAMPL8-15_micro000_c0.mol2
│ ├── SAMPL8-15_micro001_c0.mol2
│ ├── SAMPL8-15_micro002_c0.mol2
│ ├── SAMPL8-15_micro003_c0.mol2
│ ├── SAMPL8-15_micro004_c0.mol2
│ ├── SAMPL8-16_extra002_c0.mol2
│ ├── SAMPL8-16_extra003_c0.mol2
│ ├── SAMPL8-16_extra004_c0.mol2
│ ├── SAMPL8-16_extra005_c0.mol2
│ ├── SAMPL8-16_micro000_c0.mol2
│ ├── SAMPL8-16_micro004_c0.mol2
│ ├── SAMPL8-16_micro007_c0.mol2
│ ├── SAMPL8-16_micro008_c0.mol2
│ ├── SAMPL8-16_micro011_c0.mol2
│ ├── SAMPL8-17_micro000_c0.mol2
│ ├── SAMPL8-17_micro001_c0.mol2
│ ├── SAMPL8-17_micro002_c0.mol2
│ ├── SAMPL8-17_micro003_c0.mol2
│ ├── SAMPL8-17_micro004_c0.mol2
│ ├── SAMPL8-18_extra001_c0.mol2
│ ├── SAMPL8-18_micro000_c0.mol2
│ ├── SAMPL8-18_micro001_c0.mol2
│ ├── SAMPL8-18_micro002_c0.mol2
│ ├── SAMPL8-18_micro003_c0.mol2
│ ├── SAMPL8-18_micro004_c0.mol2
│ ├── SAMPL8-18_micro005_c0.mol2
│ ├── SAMPL8-19_extra001_c0.mol2
│ ├── SAMPL8-19_extra002_c0.mol2
│ ├── SAMPL8-19_extra003_c0.mol2
│ ├── SAMPL8-19_micro000_c0.mol2
│ ├── SAMPL8-19_micro002_c0.mol2
│ ├── SAMPL8-19_micro003_c0.mol2
│ ├── SAMPL8-19_micro004_c0.mol2
│ ├── SAMPL8-19_micro005_c0.mol2
│ ├── SAMPL8-19_micro006_c0.mol2
│ ├── SAMPL8-19_micro007_c0.mol2
│ ├── SAMPL8-19_micro008_c0.mol2
│ ├── SAMPL8-19_micro009_c0.mol2
│ ├── SAMPL8-19_micro010_c0.mol2
│ ├── SAMPL8-19_micro011_c0.mol2
│ ├── SAMPL8-19_micro013_c0.mol2
│ ├── SAMPL8-19_micro015_c0.mol2
│ ├── SAMPL8-19_micro017_c0.mol2
│ ├── SAMPL8-19_micro019_c0.mol2
│ ├── SAMPL8-19_micro020_c0.mol2
│ ├── SAMPL8-19_micro022_c0.mol2
│ ├── SAMPL8-19_micro024_c0.mol2
│ ├── SAMPL8-19_micro025_c0.mol2
│ ├── SAMPL8-1_extra001_c0.mol2
│ ├── SAMPL8-1_extra002_c0.mol2
│ ├── SAMPL8-1_micro000_c0.mol2
│ ├── SAMPL8-1_micro004_c0.mol2
│ ├── SAMPL8-1_micro007_c0.mol2
│ ├── SAMPL8-1_micro010_c0.mol2
│ ├── SAMPL8-20_extra001_c0.mol2
│ ├── SAMPL8-20_extra002_c0.mol2
│ ├── SAMPL8-20_extra003_c0.mol2
│ ├── SAMPL8-20_micro000_c0.mol2
│ ├── SAMPL8-20_micro001_c0.mol2
│ ├── SAMPL8-20_micro002_c0.mol2
│ ├── SAMPL8-20_micro003_c0.mol2
│ ├── SAMPL8-20_micro006_c0.mol2
│ ├── SAMPL8-20_micro011_c0.mol2
│ ├── SAMPL8-20_micro015_c0.mol2
│ ├── SAMPL8-20_micro016_c0.mol2
│ ├── SAMPL8-20_micro017_c0.mol2
│ ├── SAMPL8-20_micro018_c0.mol2
│ ├── SAMPL8-20_micro022_c0.mol2
│ ├── SAMPL8-20_micro026_c0.mol2
│ ├── SAMPL8-21_extra001_c0.mol2
│ ├── SAMPL8-21_extra002_c0.mol2
│ ├── SAMPL8-21_extra003_c0.mol2
│ ├── SAMPL8-21_extra004_c0.mol2
│ ├── SAMPL8-21_extra005_c0.mol2
│ ├── SAMPL8-21_extra006_c0.mol2
│ ├── SAMPL8-21_extra007_c0.mol2
│ ├── SAMPL8-21_extra008_c0.mol2
│ ├── SAMPL8-21_extra009_c0.mol2
│ ├── SAMPL8-21_extra010_c0.mol2
│ ├── SAMPL8-21_extra011_c0.mol2
│ ├── SAMPL8-21_extra012_c0.mol2
│ ├── SAMPL8-21_micro000_c0.mol2
│ ├── SAMPL8-21_micro004_c0.mol2
│ ├── SAMPL8-21_micro005_c0.mol2
│ ├── SAMPL8-21_micro007_c0.mol2
│ ├── SAMPL8-21_micro008_c0.mol2
│ ├── SAMPL8-21_micro009_c0.mol2
│ ├── SAMPL8-21_micro012_c0.mol2
│ ├── SAMPL8-21_micro013_c0.mol2
│ ├── SAMPL8-21_micro015_c0.mol2
│ ├── SAMPL8-21_micro016_c0.mol2
│ ├── SAMPL8-21_micro018_c0.mol2
│ ├── SAMPL8-21_micro020_c0.mol2
│ ├── SAMPL8-21_micro022_c0.mol2
│ ├── SAMPL8-21_micro023_c0.mol2
│ ├── SAMPL8-21_micro024_c0.mol2
│ ├── SAMPL8-21_micro025_c0.mol2
│ ├── SAMPL8-21_micro026_c0.mol2
│ ├── SAMPL8-21_micro027_c0.mol2
│ ├── SAMPL8-21_micro028_c0.mol2
│ ├── SAMPL8-21_micro029_c0.mol2
│ ├── SAMPL8-22_extra001_c0.mol2
│ ├── SAMPL8-22_extra002_c0.mol2
│ ├── SAMPL8-22_extra003_c0.mol2
│ ├── SAMPL8-22_extra004_c0.mol2
│ ├── SAMPL8-22_micro000_c0.mol2
│ ├── SAMPL8-22_micro001_c0.mol2
│ ├── SAMPL8-22_micro002_c0.mol2
│ ├── SAMPL8-22_micro003_c0.mol2
│ ├── SAMPL8-23_micro000_c0.mol2
│ ├── SAMPL8-23_micro002_c0.mol2
│ ├── SAMPL8-23_micro003_c0.mol2
│ ├── SAMPL8-23_micro005_c0.mol2
│ ├── SAMPL8-23_micro006_c0.mol2
│ ├── SAMPL8-23_micro007_c0.mol2
│ ├── SAMPL8-2_micro000_c0.mol2
│ ├── SAMPL8-2_micro001_c0.mol2
│ ├── SAMPL8-2_micro002_c0.mol2
│ ├── SAMPL8-3_extra001_c0.mol2
│ ├── SAMPL8-3_extra002_c0.mol2
│ ├── SAMPL8-3_extra003_c0.mol2
│ ├── SAMPL8-3_micro000_c0.mol2
│ ├── SAMPL8-3_micro006_c0.mol2
│ ├── SAMPL8-3_micro010_c0.mol2
│ ├── SAMPL8-3_micro013_c0.mol2
│ ├── SAMPL8-3_micro016_c0.mol2
│ ├── SAMPL8-4_extra001_c0.mol2
│ ├── SAMPL8-4_extra002_c0.mol2
│ ├── SAMPL8-4_micro000_c0.mol2
│ ├── SAMPL8-4_micro001_c0.mol2
│ ├── SAMPL8-4_micro002_c0.mol2
│ ├── SAMPL8-4_micro003_c0.mol2
│ ├── SAMPL8-4_micro005_c0.mol2
│ ├── SAMPL8-4_micro008_c0.mol2
│ ├── SAMPL8-4_micro010_c0.mol2
│ ├── SAMPL8-5_micro000_c0.mol2
│ ├── SAMPL8-5_micro001_c0.mol2
│ ├── SAMPL8-5_micro003_c0.mol2
│ ├── SAMPL8-5_micro005_c0.mol2
│ ├── SAMPL8-5_micro006_c0.mol2
│ ├── SAMPL8-5_micro007_c0.mol2
│ ├── SAMPL8-6_micro000_c0.mol2
│ ├── SAMPL8-6_micro001_c0.mol2
│ ├── SAMPL8-6_micro003_c0.mol2
│ ├── SAMPL8-6_micro007_c0.mol2
│ ├── SAMPL8-6_micro009_c0.mol2
│ ├── SAMPL8-7_micro000_c0.mol2
│ ├── SAMPL8-7_micro001_c0.mol2
│ ├── SAMPL8-7_micro002_c0.mol2
│ ├── SAMPL8-7_micro003_c0.mol2
│ ├── SAMPL8-7_micro004_c0.mol2
│ ├── SAMPL8-8_micro000_c0.mol2
│ ├── SAMPL8-8_micro001_c0.mol2
│ ├── SAMPL8-8_micro002_c0.mol2
│ ├── SAMPL8-9_micro000_c0.mol2
│ ├── SAMPL8-9_micro001_c0.mol2
│ ├── SAMPL8-9_micro002_c0.mol2
│ ├── SAMPL8-9_micro003_c0.mol2
│ └── SAMPL8-9_micro004_c0.mol2
├── dortmund_microstates
│ ├── SAMPL8-1
│ │ └── extra001
│ │ │ └── mmopt.mol2
│ ├── SAMPL8-12
│ │ ├── extra001
│ │ │ └── mmopt.mol2
│ │ ├── extra002
│ │ │ └── mmopt.mol2
│ │ ├── extra003
│ │ │ └── mmopt.mol2
│ │ ├── extra004
│ │ │ └── mmopt.mol2
│ │ ├── extra005
│ │ │ └── mmopt.mol2
│ │ └── extra006
│ │ │ └── mmopt.mol2
│ ├── SAMPL8-14
│ │ ├── extra001
│ │ │ └── mmopt.mol2
│ │ ├── extra002
│ │ │ └── mmopt.mol2
│ │ ├── extra003
│ │ │ └── mmopt.mol2
│ │ ├── extra004
│ │ │ └── mmopt.mol2
│ │ ├── extra005
│ │ │ └── mmopt.mol2
│ │ ├── extra006
│ │ │ └── mmopt.mol2
│ │ ├── extra007
│ │ │ └── mmopt.mol2
│ │ ├── extra008
│ │ │ └── mmopt.mol2
│ │ ├── extra009
│ │ │ └── mmopt.mol2
│ │ ├── extra010
│ │ │ └── mmopt.mol2
│ │ ├── extra011
│ │ │ └── mmopt.mol2
│ │ └── extra012
│ │ │ └── mmopt.mol2
│ ├── SAMPL8-21
│ │ ├── extra001
│ │ │ └── mmopt.mol2
│ │ ├── extra002
│ │ │ └── mmopt.mol2
│ │ ├── extra003
│ │ │ └── mmopt.mol2
│ │ ├── extra004
│ │ │ └── mmopt.mol2
│ │ ├── extra005
│ │ │ └── mmopt.mol2
│ │ ├── extra006
│ │ │ └── mmopt.mol2
│ │ ├── extra007
│ │ │ └── mmopt.mol2
│ │ ├── extra008
│ │ │ └── mmopt.mol2
│ │ ├── extra009
│ │ │ └── mmopt.mol2
│ │ ├── extra010
│ │ │ └── mmopt.mol2
│ │ └── extra011
│ │ │ └── mmopt.mol2
│ ├── SAMPL8-22
│ │ ├── extra001
│ │ │ └── mmopt.mol2
│ │ ├── extra002
│ │ │ └── mmopt.mol2
│ │ ├── extra003
│ │ │ └── mmopt.mol2
│ │ ├── extra004
│ │ │ └── mmopt.mol2
│ │ └── extra005
│ │ │ └── mmopt.mol2
│ └── SAMPL8-3
│ │ └── extra001
│ │ └── mmopt.mol2
└── make_mol2_sdf_pdb_files.ipynb
├── pKa
├── README.md
├── SAMPL8-pKa-user-map.csv
├── example_submission_file
│ ├── PKA_submission.csv
│ └── example_submission.csv
├── experimental_pKas.csv
├── macrostate_analysis
│ ├── README.md
│ ├── Titration_Curves.pdf
│ ├── functions_pKa_macrostate_analysis.py
│ ├── pKa_macrostate_analysis_popular_transitions.py
│ ├── pKa_macrostate_analysis_selected_transitions.py
│ ├── popular_transitions_analysis
│ │ ├── README.md
│ │ ├── analysis_outputs_all
│ │ │ ├── Correlation_Plots
│ │ │ │ ├── Correlation_statistics.csv
│ │ │ │ ├── PKA_ECRISMCorr_plot.pdf
│ │ │ │ ├── pKa-3DS-1Corr_plot.pdf
│ │ │ │ ├── pKa-3DS-2Corr_plot.pdf
│ │ │ │ ├── pKa-3DS-3Corr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_AdaBoostCorr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_DeepGPCorr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_RFCorr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_XGBoostCorr_plot.pdf
│ │ │ │ ├── pKa-ZhiyiWu-1Corr_plot.pdf
│ │ │ │ ├── pKa_ChemaxonCorr_plot.pdf
│ │ │ │ ├── pKa_SabatinoRodriguezPaluch_uESECorr_plot.pdf
│ │ │ │ └── pKa_SabatinoRodriguezPaluch_uESE_extraCorr_plot.pdf
│ │ │ ├── Error_statistics.csv
│ │ │ ├── README.md
│ │ │ ├── abs_error_bymethod_plot.pdf
│ │ │ ├── abs_error_bymol_plot.pdf
│ │ │ ├── macrostate_pKa_data.csv
│ │ │ ├── mean_abs_error_plot.pdf
│ │ │ ├── mean_error_plot.pdf
│ │ │ ├── popular_transitions_pKa_data.csv
│ │ │ └── rmse_plot.pdf
│ │ └── analysis_outputs_ranked
│ │ │ ├── Correlation_Plots
│ │ │ ├── Correlation_statistics.csv
│ │ │ ├── PKA_ECRISMCorr_plot.pdf
│ │ │ ├── pKa-3DS-1Corr_plot.pdf
│ │ │ ├── pKa-RobertRaddi_DeepGPCorr_plot.pdf
│ │ │ ├── pKa-ZhiyiWu-1Corr_plot.pdf
│ │ │ ├── pKa_ChemaxonCorr_plot.pdf
│ │ │ └── pKa_SabatinoRodriguezPaluch_uESE_extraCorr_plot.pdf
│ │ │ ├── Error_statistics.csv
│ │ │ ├── README.md
│ │ │ ├── abs_error_bymethod_plot.pdf
│ │ │ ├── abs_error_bymol_plot.pdf
│ │ │ ├── macrostate_pKa_data.csv
│ │ │ ├── mean_abs_error_plot.pdf
│ │ │ ├── mean_error_plot.pdf
│ │ │ ├── popular_transitions_pKa_data.csv
│ │ │ └── rmse_plot.pdf
│ ├── selected_transitions.csv
│ ├── selected_transitions_analysis
│ │ ├── README.md
│ │ ├── analysis_outputs_all
│ │ │ ├── Correlation_Plots
│ │ │ │ ├── Correlation_statistics.csv
│ │ │ │ ├── PKA_ECRISMCorr_plot.pdf
│ │ │ │ ├── pKa-3DS-1Corr_plot.pdf
│ │ │ │ ├── pKa-3DS-2Corr_plot.pdf
│ │ │ │ ├── pKa-3DS-3Corr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_AdaBoostCorr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_DeepGPCorr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_RFCorr_plot.pdf
│ │ │ │ ├── pKa-RobertRaddi_XGBoostCorr_plot.pdf
│ │ │ │ ├── pKa-ZhiyiWu-1Corr_plot.pdf
│ │ │ │ ├── pKa_ChemaxonCorr_plot.pdf
│ │ │ │ ├── pKa_SabatinoRodriguezPaluch_uESECorr_plot.pdf
│ │ │ │ └── pKa_SabatinoRodriguezPaluch_uESE_extraCorr_plot.pdf
│ │ │ ├── Error_statistics.csv
│ │ │ ├── abs_error_bymethod_plot.pdf
│ │ │ ├── abs_error_bymol_plot.pdf
│ │ │ ├── macrostate_pKa_data.csv
│ │ │ ├── mean_abs_error_plot.pdf
│ │ │ ├── mean_error_plot.pdf
│ │ │ ├── popular_transitions_pKa_data.csv
│ │ │ └── rmse_plot.pdf
│ │ └── analysis_outputs_ranked
│ │ │ ├── Correlation_Plots
│ │ │ ├── Correlation_statistics.csv
│ │ │ ├── PKA_ECRISMCorr_plot.pdf
│ │ │ ├── pKa-3DS-1Corr_plot.pdf
│ │ │ ├── pKa-RobertRaddi_DeepGPCorr_plot.pdf
│ │ │ ├── pKa-ZhiyiWu-1Corr_plot.pdf
│ │ │ ├── pKa_ChemaxonCorr_plot.pdf
│ │ │ └── pKa_SabatinoRodriguezPaluch_uESE_extraCorr_plot.pdf
│ │ │ ├── Error_statistics.csv
│ │ │ ├── abs_error_bymethod_plot.pdf
│ │ │ ├── abs_error_bymol_plot.pdf
│ │ │ ├── macrostate_pKa_data.csv
│ │ │ ├── mean_abs_error_plot.pdf
│ │ │ ├── mean_error_plot.pdf
│ │ │ ├── popular_transitions_pKa_data.csv
│ │ │ └── rmse_plot.pdf
│ ├── titration_curve_plots
│ │ ├── PKA_ECRISM:SAMPL8-1.pdf
│ │ ├── PKA_ECRISM:SAMPL8-10.pdf
│ │ ├── PKA_ECRISM:SAMPL8-12.pdf
│ │ ├── PKA_ECRISM:SAMPL8-14.pdf
│ │ ├── PKA_ECRISM:SAMPL8-15.pdf
│ │ ├── PKA_ECRISM:SAMPL8-16.pdf
│ │ ├── PKA_ECRISM:SAMPL8-17.pdf
│ │ ├── PKA_ECRISM:SAMPL8-18.pdf
│ │ ├── PKA_ECRISM:SAMPL8-19.pdf
│ │ ├── PKA_ECRISM:SAMPL8-2.pdf
│ │ ├── PKA_ECRISM:SAMPL8-20.pdf
│ │ ├── PKA_ECRISM:SAMPL8-21.pdf
│ │ ├── PKA_ECRISM:SAMPL8-22.pdf
│ │ ├── PKA_ECRISM:SAMPL8-23.pdf
│ │ ├── PKA_ECRISM:SAMPL8-3.pdf
│ │ ├── PKA_ECRISM:SAMPL8-4.pdf
│ │ ├── PKA_ECRISM:SAMPL8-5.pdf
│ │ ├── PKA_ECRISM:SAMPL8-6.pdf
│ │ ├── PKA_ECRISM:SAMPL8-7.pdf
│ │ ├── PKA_ECRISM:SAMPL8-8.pdf
│ │ ├── PKA_ECRISM:SAMPL8-9.pdf
│ │ ├── macro_pKas_data.csv
│ │ ├── pKa-3DS-1:SAMPL8-1.pdf
│ │ ├── pKa-3DS-1:SAMPL8-10.pdf
│ │ ├── pKa-3DS-1:SAMPL8-12.pdf
│ │ ├── pKa-3DS-1:SAMPL8-14.pdf
│ │ ├── pKa-3DS-1:SAMPL8-15.pdf
│ │ ├── pKa-3DS-1:SAMPL8-16.pdf
│ │ ├── pKa-3DS-1:SAMPL8-17.pdf
│ │ ├── pKa-3DS-1:SAMPL8-18.pdf
│ │ ├── pKa-3DS-1:SAMPL8-19.pdf
│ │ ├── pKa-3DS-1:SAMPL8-2.pdf
│ │ ├── pKa-3DS-1:SAMPL8-20.pdf
│ │ ├── pKa-3DS-1:SAMPL8-21.pdf
│ │ ├── pKa-3DS-1:SAMPL8-22.pdf
│ │ ├── pKa-3DS-1:SAMPL8-23.pdf
│ │ ├── pKa-3DS-1:SAMPL8-3.pdf
│ │ ├── pKa-3DS-1:SAMPL8-4.pdf
│ │ ├── pKa-3DS-1:SAMPL8-5.pdf
│ │ ├── pKa-3DS-1:SAMPL8-6.pdf
│ │ ├── pKa-3DS-1:SAMPL8-7.pdf
│ │ ├── pKa-3DS-1:SAMPL8-8.pdf
│ │ ├── pKa-3DS-1:SAMPL8-9.pdf
│ │ ├── pKa-3DS-2:SAMPL8-1.pdf
│ │ ├── pKa-3DS-2:SAMPL8-10.pdf
│ │ ├── pKa-3DS-2:SAMPL8-12.pdf
│ │ ├── pKa-3DS-2:SAMPL8-14.pdf
│ │ ├── pKa-3DS-2:SAMPL8-15.pdf
│ │ ├── pKa-3DS-2:SAMPL8-16.pdf
│ │ ├── pKa-3DS-2:SAMPL8-17.pdf
│ │ ├── pKa-3DS-2:SAMPL8-18.pdf
│ │ ├── pKa-3DS-2:SAMPL8-19.pdf
│ │ ├── pKa-3DS-2:SAMPL8-2.pdf
│ │ ├── pKa-3DS-2:SAMPL8-20.pdf
│ │ ├── pKa-3DS-2:SAMPL8-21.pdf
│ │ ├── pKa-3DS-2:SAMPL8-22.pdf
│ │ ├── pKa-3DS-2:SAMPL8-23.pdf
│ │ ├── pKa-3DS-2:SAMPL8-3.pdf
│ │ ├── pKa-3DS-2:SAMPL8-4.pdf
│ │ ├── pKa-3DS-2:SAMPL8-5.pdf
│ │ ├── pKa-3DS-2:SAMPL8-6.pdf
│ │ ├── pKa-3DS-2:SAMPL8-7.pdf
│ │ ├── pKa-3DS-2:SAMPL8-8.pdf
│ │ ├── pKa-3DS-2:SAMPL8-9.pdf
│ │ ├── pKa-3DS-3:SAMPL8-1.pdf
│ │ ├── pKa-3DS-3:SAMPL8-10.pdf
│ │ ├── pKa-3DS-3:SAMPL8-12.pdf
│ │ ├── pKa-3DS-3:SAMPL8-14.pdf
│ │ ├── pKa-3DS-3:SAMPL8-15.pdf
│ │ ├── pKa-3DS-3:SAMPL8-16.pdf
│ │ ├── pKa-3DS-3:SAMPL8-17.pdf
│ │ ├── pKa-3DS-3:SAMPL8-18.pdf
│ │ ├── pKa-3DS-3:SAMPL8-19.pdf
│ │ ├── pKa-3DS-3:SAMPL8-2.pdf
│ │ ├── pKa-3DS-3:SAMPL8-20.pdf
│ │ ├── pKa-3DS-3:SAMPL8-21.pdf
│ │ ├── pKa-3DS-3:SAMPL8-22.pdf
│ │ ├── pKa-3DS-3:SAMPL8-23.pdf
│ │ ├── pKa-3DS-3:SAMPL8-3.pdf
│ │ ├── pKa-3DS-3:SAMPL8-4.pdf
│ │ ├── pKa-3DS-3:SAMPL8-5.pdf
│ │ ├── pKa-3DS-3:SAMPL8-6.pdf
│ │ ├── pKa-3DS-3:SAMPL8-7.pdf
│ │ ├── pKa-3DS-3:SAMPL8-8.pdf
│ │ ├── pKa-3DS-3:SAMPL8-9.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-1.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-10.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-12.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-14.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-15.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-16.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-17.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-18.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-19.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-2.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-20.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-21.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-22.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-23.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-3.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-4.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-5.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-6.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-7.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-8.pdf
│ │ ├── pKa-RobertRaddi_AdaBoost:SAMPL8-9.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-1.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-10.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-12.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-14.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-15.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-16.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-17.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-18.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-19.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-2.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-20.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-21.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-22.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-23.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-3.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-4.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-5.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-6.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-7.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-8.pdf
│ │ ├── pKa-RobertRaddi_DeepGP:SAMPL8-9.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-1.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-10.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-12.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-14.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-15.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-16.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-17.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-18.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-19.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-2.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-20.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-21.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-22.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-23.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-3.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-4.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-5.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-6.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-7.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-8.pdf
│ │ ├── pKa-RobertRaddi_RF:SAMPL8-9.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-1.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-10.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-12.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-14.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-15.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-16.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-17.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-18.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-19.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-2.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-20.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-21.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-22.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-23.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-3.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-4.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-5.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-6.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-7.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-8.pdf
│ │ ├── pKa-RobertRaddi_XGBoost:SAMPL8-9.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-1.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-10.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-12.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-14.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-15.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-16.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-17.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-18.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-19.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-2.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-20.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-21.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-22.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-23.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-3.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-4.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-5.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-6.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-7.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-8.pdf
│ │ ├── pKa-ZhiyiWu-1:SAMPL8-9.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-1.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-10.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-12.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-14.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-15.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-16.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-17.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-18.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-19.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-2.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-20.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-21.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-22.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-23.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-3.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-4.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-5.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-6.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-7.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-8.pdf
│ │ ├── pKa_Chemaxon:SAMPL8-9.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-1.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-10.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-12.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-14.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-15.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-16.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-17.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-18.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-19.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-2.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-20.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-21.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-22.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-23.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-3.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-4.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-5.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-6.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-7.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-8.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE:SAMPL8-9.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-1.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-10.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-12.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-14.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-15.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-16.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-17.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-18.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-19.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-2.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-20.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-21.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-22.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-23.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-3.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-4.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-5.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-6.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-7.pdf
│ │ ├── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-8.pdf
│ │ └── pKa_SabatinoRodriguezPaluch_uESE_extra:SAMPL8-9.pdf
│ └── titration_curves.py
├── pKa_challenge_instructions.md
├── relative_microstate_free_energy_predictions
│ ├── PKA_ECRISM.csv
│ ├── README.md
│ ├── pKa-3DS-1.csv
│ ├── pKa-3DS-2.csv
│ ├── pKa-3DS-3.csv
│ ├── pKa-RobertRaddi_AdaBoost.csv
│ ├── pKa-RobertRaddi_DeepGP.csv
│ ├── pKa-RobertRaddi_RF.csv
│ ├── pKa-RobertRaddi_XGBoost.csv
│ ├── pKa-ZhiyiWu-1.csv
│ ├── pKa_Chemaxon.csv
│ ├── pKa_SabatinoRodriguezPaluch_uESE.csv
│ └── pKa_SabatinoRodriguezPaluch_uESE_extra.csv
├── submission_template_file
│ └── pKa_prediction_template.csv
└── submissions
│ ├── PKA_ECRISM.csv
│ ├── README.md
│ ├── pKa-3DS-1.csv
│ ├── pKa-3DS-2.csv
│ ├── pKa-3DS-3.csv
│ ├── pKa-RobertRaddi_AdaBoost.csv
│ ├── pKa-RobertRaddi_DeepGP.csv
│ ├── pKa-RobertRaddi_RF.csv
│ ├── pKa-RobertRaddi_XGBoost.csv
│ ├── pKa-ZhiyiWu-1.csv
│ ├── pKa_Chemaxon.csv
│ ├── pKa_SabatinoRodriguezPaluch_uESE.csv
│ └── pKa_SabatinoRodriguezPaluch_uESE_extra.csv
└── source_data
├── compounds.pdf
├── compounds.pptx
└── ~$compounds.pptx
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1 | #!/usr/bin/env python
2 |
3 | """Analysis code for the SAMPL and SAMPLing challenges."""
4 |
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1 | Methamphetamine;G1
2 | Fentanyl;G2
3 | Morphine;G3
4 | Hydromorphone;G4
5 | Ketamine;G5
6 | PhenylCyclohexylPiperidine(PCP);G6
7 | Cocaine;G7
8 |
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1 | microstate ID,canonical isomeric SMILES
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3 | SAMPL8-10_micro001,CS(=O)(=O)c1cccc(c1)c2ccc(cc2)C[NH2+]Cc3c(cccc3Cl)F
4 |
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3 | SAMPL8-13_micro001,C[C@H](c1ccccc1Cl)Oc2cc(sc2C(=O)N)n3c[nH+]c4c3cc(cc4)S(=O)(=O)C
4 | SAMPL8-13_micro002,C[C@@H](Oc1cc(sc1C([NH-])=O)-n1cnc2ccc(cc12)S(C)(=O)=O)c1ccccc1Cl
5 |
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3 | SAMPL8-2_micro001,CS(=O)(=O)c1ccc(cc1)CCC(=O)[O-]
4 | SAMPL8-2_micro002,CS(=O)(=O)c1ccc(cc1)CC=C(O)O
5 | SAMPL8-2_micro003,CS(=O)(=O)c1ccc(cc1)CC=C(O)[O-]
6 |
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1 | microstate ID,canonical isomeric SMILES
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3 | SAMPL8-8_micro001,COC(=C1C=[n+]2cccc(c2=[NH+]1)C(F)(F)F)[O-]
4 | SAMPL8-8_micro002,COC(=C1C=[n+]2cccc(c2=N1)C(F)(F)F)O
5 |
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1 | David Mobley D a v i d M o b l e y
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